6.1 Introduction6.2 Basolateral Transporters6.3 Canalicular Transporters6.4 Data Sources for Transporters in Hepatotoxicity6.5 In Silico Transporters Models6.6 Ligand-Based Approaches6.7 OATP1B1 and OATP1B36.8 NTCP6.9 OCT16.10 OCT26.11 MRP1, MRP3, and MRP46.12 BSEP6.13 MRP26.14 MDR1/P-gp6.15 MDR36.16 BCRP6.17 MATE16.18 ASBT6.19 Structure-Based Approaches6.20 Complex Models Incorporating Transporter Information6.21 In Vitro Models6.22 Multiscale Models6.23 OutlookAcknowledgmentsReferences